2:00 Assessing Bifunctional Protein Degraders for Oral Delivery
Time: 9:30 am
day: Day 1 Track A morning
Details:
- Understand why bifunctional protein degraders cannot be evaluated through a conventional small molecule lens
- Explore the key physicochemical properties that determine whether a bifunctional protein degrader is likely to be orally bioavailable
- Discuss rate limiting steps to oral absorption and how enabling technologies may enhance absorption of this class of molecule
