Harnessing AI & Structural Proteomics for Rational Computational Design of Degraders

  • Demonstrating how the AIMS (AI + MS) platform integrates AI modelling and structural proteomics to map protein interactions and inform degrader design
  • Showcasing lead optimisation strategies to enhance efficacy, selectivity, and rational design of molecular glues and degraders
  • Presenting preclinical results from Protai’s KAT6 degrader program as a case study of AIMS enabled design