Harnessing AI & Structural Proteomics to Drive Rational Design and Lead Optimisation in Molecular Glue & Degrader Discovery
- Demonstrating how the AIMS (AI + MS) platform integrates AI modelling and structural proteomics to map protein interactions and inform degrader design
- Showcasing lead optimisation strategies to enhance efficacy, selectivity, and rational design of molecular glues and degraders
- Presenting preclinical results from Protai’s CAR-T6 degrader program as a case study of data-driven optimisation from discovery to in vivo validation